Ligand source activities (1 row/activity)



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Ligands (move mouse cursor over ligand name to see structure) Receptor Assay information Chemical information
Sel. page Common
name		 GPCRdb
ID		 #Vendors

 Reference
ligand		 Fold
selectivity		 # Tested
GPCRs		 Species

 p-value
(-log)		 Activity
Type		 Activity
Relation		 Activity
Value		 AssayType

 Assay
Description		 Source

 Mol
weight		 Rot
Bonds		 H don

 H acc

 LogP

 Smiles

 DOI
131648253 3039 0 None - 1 Mouse 10.7 pEC50 = 10.7 Functional
High affinity binding site of mouse GPR83High affinity binding site of mouse GPR83
Guide to Pharmacology None None None None 27117253
155817507 3039 0 None - 1 Mouse 10.7 pEC50 = 10.7 Functional
High affinity binding site of mouse GPR83High affinity binding site of mouse GPR83
Guide to Pharmacology None None None None 27117253
9139 3039 0 None - 1 Mouse 10.7 pEC50 = 10.7 Functional
High affinity binding site of mouse GPR83High affinity binding site of mouse GPR83
Guide to Pharmacology None None None None 27117253
131648253 3039 0 None - 1 Mouse 7.0 pEC50 = 7.0 Functional
Low affinity binding site of mouse GPR83Low affinity binding site of mouse GPR83
Guide to Pharmacology None None None None 27117253
155817507 3039 0 None - 1 Mouse 7.0 pEC50 = 7.0 Functional
Low affinity binding site of mouse GPR83Low affinity binding site of mouse GPR83
Guide to Pharmacology None None None None 27117253
9139 3039 0 None - 1 Mouse 7.0 pEC50 = 7.0 Functional
Low affinity binding site of mouse GPR83Low affinity binding site of mouse GPR83
Guide to Pharmacology None None None None 27117253
32051 4151 0 None - 1 Mouse 5.0 pEC50 = 5 Functional
UnclassifiedUnclassified
Guide to Pharmacology 64 0 0 0 -0.0 [Zn+2] 23335960
566 4151 0 None - 1 Mouse 5.0 pEC50 = 5 Functional
UnclassifiedUnclassified
Guide to Pharmacology 64 0 0 0 -0.0 [Zn+2] 23335960


Get vendors


Ligands (move mouse cursor over ligand name to see structure) Receptor Assay information Chemical information
Sel. page Similar-
ity		 Common
name		 GPCRdb
ID		 #Vendors

 Reference
ligand		 Fold
selectivity		 # Tested
GPCRs		 Species

 p-value
(-log)		 Activity
Type		 Activity
Relation		 Activity
Value		 Assay
Type		 Assay
Description		 Source

 Mol
weight		 Rot
Bonds		 H don

 H acc

 LogP

 Smiles

 DOI
9140 3040 0 None - 1 Mouse 8.1 pKd = 8.1 Binding
N-terminally tyrosinated radioidodinated rPEN binding to mouse GPR83 in hypothalamic membrane preparations.N-terminally tyrosinated radioidodinated rPEN binding to mouse GPR83 in hypothalamic membrane preparations.
Guide to Pharmacology None None None None 27117253