Ligand source activities (1 row/activity)
| Ligands (move mouse cursor over ligand name to see structure) | Receptor | Assay information | Chemical information | ||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Sel. page | Common name
| GPCRdb ID
| #Vendors | Reference ligand
| Fold selectivity | # Tested GPCRs | Species
| p-value (-log) | Activity Type
| Activity Relation
| Activity Value
| AssayType
| Assay Description
| Source
| Mol weight | Rot Bonds | H don | H acc | LogP | Smiles
| DOI
|
Ligands (move mouse cursor over ligand name to see structure)
| Receptor
| Assay information
| Chemical information
| ||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sel. page | Common name
| GPCRdb ID
| #Vendors | Reference ligand
| Fold selectivity | # Tested GPCRs | Species
| p-value (-log) | Activity Type
| Activity Relation
| Activity Value
| AssayType
| Assay Description
| Source
| Mol weight | Rot Bonds | H don | H acc | LogP | Smiles
| DOI
|
| 5572 | 1928 | 0 | None | - | 1 | Rat | 7.6 | pA2 | = | 7.6 | Functional | UnclassifiedUnclassified |
Guide to Pharmacology | None | None | None | None | None | |||
| 129631922 | 3781 | 13 | None | -34 | 4 | Rat | 8.2 | pIC50 | = | 8.2 | Functional | NoneNone |
Drug Central | None | None | None | None | None | |||
| 132274287 | 3781 | 13 | None | -34 | 4 | Rat | 8.2 | pIC50 | = | 8.2 | Functional | NoneNone |
Drug Central | None | None | None | None | None | |||
| 132451761 | 3781 | 13 | None | -34 | 4 | Rat | 8.2 | pIC50 | = | 8.2 | Functional | NoneNone |
Drug Central | None | None | None | None | None | |||
| 155817470 | 3781 | 13 | None | -34 | 4 | Rat | 8.2 | pIC50 | = | 8.2 | Functional | NoneNone |
Drug Central | None | None | None | None | None | |||
| 16132393 | 3781 | 13 | None | -34 | 4 | Rat | 8.2 | pIC50 | = | 8.2 | Functional | NoneNone |
Drug Central | None | None | None | None | None | |||
| 16133850 | 3781 | 13 | None | -34 | 4 | Rat | 8.2 | pIC50 | = | 8.2 | Functional | NoneNone |
Drug Central | None | None | None | None | None | |||
| 4448 | 3781 | 13 | None | -34 | 4 | Rat | 8.2 | pIC50 | = | 8.2 | Functional | NoneNone |
Drug Central | None | None | None | None | None | |||
| 4514 | 3781 | 13 | None | -34 | 4 | Rat | 8.2 | pIC50 | = | 8.2 | Functional | NoneNone |
Drug Central | None | None | None | None | None | |||
| 91933454 | 3781 | 13 | None | -34 | 4 | Rat | 8.2 | pIC50 | = | 8.2 | Functional | NoneNone |
Drug Central | None | None | None | None | None | |||
| CHEMBL525610 | 3781 | 13 | None | -34 | 4 | Rat | 8.2 | pIC50 | = | 8.2 | Functional | NoneNone |
Drug Central | None | None | None | None | None | |||
| DB06285 | 3781 | 13 | None | -34 | 4 | Rat | 8.2 | pIC50 | = | 8.2 | Functional | NoneNone |
Drug Central | None | None | None | None | None | |||
| 129631922 | 3781 | 13 | None | -7 | 4 | Human | 8.1 | pIC50 | = | 8.1 | Functional | NoneNone |
Drug Central | None | None | None | None | None | |||
| 132274287 | 3781 | 13 | None | -7 | 4 | Human | 8.1 | pIC50 | = | 8.1 | Functional | NoneNone |
Drug Central | None | None | None | None | None | |||
| 132451761 | 3781 | 13 | None | -7 | 4 | Human | 8.1 | pIC50 | = | 8.1 | Functional | NoneNone |
Drug Central | None | None | None | None | None | |||
| 155817470 | 3781 | 13 | None | -7 | 4 | Human | 8.1 | pIC50 | = | 8.1 | Functional | NoneNone |
Drug Central | None | None | None | None | None | |||
| 16132393 | 3781 | 13 | None | -7 | 4 | Human | 8.1 | pIC50 | = | 8.1 | Functional | NoneNone |
Drug Central | None | None | None | None | None | |||
| 16133850 | 3781 | 13 | None | -7 | 4 | Human | 8.1 | pIC50 | = | 8.1 | Functional | NoneNone |
Drug Central | None | None | None | None | None | |||
| 4448 | 3781 | 13 | None | -7 | 4 | Human | 8.1 | pIC50 | = | 8.1 | Functional | NoneNone |
Drug Central | None | None | None | None | None | |||
| 4514 | 3781 | 13 | None | -7 | 4 | Human | 8.1 | pIC50 | = | 8.1 | Functional | NoneNone |
Drug Central | None | None | None | None | None | |||
| 91933454 | 3781 | 13 | None | -7 | 4 | Human | 8.1 | pIC50 | = | 8.1 | Functional | NoneNone |
Drug Central | None | None | None | None | None | |||
| CHEMBL525610 | 3781 | 13 | None | -7 | 4 | Human | 8.1 | pIC50 | = | 8.1 | Functional | NoneNone |
Drug Central | None | None | None | None | None | |||
| DB06285 | 3781 | 13 | None | -7 | 4 | Human | 8.1 | pIC50 | = | 8.1 | Functional | NoneNone |
Drug Central | None | None | None | None | None | |||
| 155817427 | 3232 | 0 | None | -158 | 3 | Rat | 5.5 | pIC50 | = | 5.5 | Functional | UnclassifiedUnclassified |
Guide to Pharmacology | None | None | None | None | 11602681 | |||
| 1788 | 3232 | 0 | None | -158 | 3 | Rat | 5.5 | pIC50 | = | 5.5 | Functional | UnclassifiedUnclassified |
Guide to Pharmacology | None | None | None | None | 11602681 | |||
| 129316189 | 3229 | 0 | None | -35 | 3 | Rat | 6.8 | pIC50 | = | 6.8 | Functional | UnclassifiedUnclassified |
Guide to Pharmacology | None | None | None | None | 11602681 | |||
| 155817471 | 3229 | 0 | None | -35 | 3 | Rat | 6.8 | pIC50 | = | 6.8 | Functional | UnclassifiedUnclassified |
Guide to Pharmacology | None | None | None | None | 11602681 | |||
| 16201228 | 3229 | 0 | None | -35 | 3 | Rat | 6.8 | pIC50 | = | 6.8 | Functional | UnclassifiedUnclassified |
Guide to Pharmacology | None | None | None | None | 11602681 | |||
| 4449 | 3229 | 0 | None | -35 | 3 | Rat | 6.8 | pIC50 | = | 6.8 | Functional | UnclassifiedUnclassified |
Guide to Pharmacology | None | None | None | None | 11602681 | |||
| 1824 | 2003 | 0 | None | - | 1 | Human | 7.0 | pIC50 | = | 7 | Functional | UnclassifiedUnclassified |
Guide to Pharmacology | None | None | None | None | 10537121 | |||
| 155817427 | 3232 | 0 | None | -1 | 3 | Human | 7.5 | pIC50 | = | 7.5 | Functional | UnclassifiedUnclassified |
Guide to Pharmacology | None | None | None | None | 11602681 | |||
| 155817427 | 3232 | 0 | None | -1 | 3 | Human | 7.5 | pIC50 | = | 7.5 | Functional | UnclassifiedUnclassified |
Guide to Pharmacology | None | None | None | None | 8702701 | |||
| 1788 | 3232 | 0 | None | -1 | 3 | Human | 7.5 | pIC50 | = | 7.5 | Functional | UnclassifiedUnclassified |
Guide to Pharmacology | None | None | None | None | 11602681 | |||
| 1788 | 3232 | 0 | None | -1 | 3 | Human | 7.5 | pIC50 | = | 7.5 | Functional | UnclassifiedUnclassified |
Guide to Pharmacology | None | None | None | None | 8702701 | |||
| 129631922 | 3781 | 13 | None | -7 | 4 | Human | 7.8 | pIC50 | = | 7.8 | Functional | UnclassifiedUnclassified |
Guide to Pharmacology | None | None | None | None | 11602681 | |||
| 129631922 | 3781 | 13 | None | -7 | 4 | Human | 7.8 | pIC50 | = | 7.8 | Functional | UnclassifiedUnclassified |
Guide to Pharmacology | None | None | None | None | 8702701 | |||
| 132274287 | 3781 | 13 | None | -7 | 4 | Human | 7.8 | pIC50 | = | 7.8 | Functional | UnclassifiedUnclassified |
Guide to Pharmacology | None | None | None | None | 11602681 | |||
| 132274287 | 3781 | 13 | None | -7 | 4 | Human | 7.8 | pIC50 | = | 7.8 | Functional | UnclassifiedUnclassified |
Guide to Pharmacology | None | None | None | None | 8702701 | |||
| 132451761 | 3781 | 13 | None | -7 | 4 | Human | 7.8 | pIC50 | = | 7.8 | Functional | UnclassifiedUnclassified |
Guide to Pharmacology | None | None | None | None | 11602681 | |||
| 132451761 | 3781 | 13 | None | -7 | 4 | Human | 7.8 | pIC50 | = | 7.8 | Functional | UnclassifiedUnclassified |
Guide to Pharmacology | None | None | None | None | 8702701 | |||
| 155817470 | 3781 | 13 | None | -7 | 4 | Human | 7.8 | pIC50 | = | 7.8 | Functional | UnclassifiedUnclassified |
Guide to Pharmacology | None | None | None | None | 11602681 | |||
| 155817470 | 3781 | 13 | None | -7 | 4 | Human | 7.8 | pIC50 | = | 7.8 | Functional | UnclassifiedUnclassified |
Guide to Pharmacology | None | None | None | None | 8702701 | |||
| 16132393 | 3781 | 13 | None | -7 | 4 | Human | 7.8 | pIC50 | = | 7.8 | Functional | UnclassifiedUnclassified |
Guide to Pharmacology | None | None | None | None | 11602681 | |||
| 16132393 | 3781 | 13 | None | -7 | 4 | Human | 7.8 | pIC50 | = | 7.8 | Functional | UnclassifiedUnclassified |
Guide to Pharmacology | None | None | None | None | 8702701 | |||
| 16133850 | 3781 | 13 | None | -7 | 4 | Human | 7.8 | pIC50 | = | 7.8 | Functional | UnclassifiedUnclassified |
Guide to Pharmacology | None | None | None | None | 11602681 | |||
| 16133850 | 3781 | 13 | None | -7 | 4 | Human | 7.8 | pIC50 | = | 7.8 | Functional | UnclassifiedUnclassified |
Guide to Pharmacology | None | None | None | None | 8702701 | |||
| 4448 | 3781 | 13 | None | -7 | 4 | Human | 7.8 | pIC50 | = | 7.8 | Functional | UnclassifiedUnclassified |
Guide to Pharmacology | None | None | None | None | 11602681 | |||
| 4448 | 3781 | 13 | None | -7 | 4 | Human | 7.8 | pIC50 | = | 7.8 | Functional | UnclassifiedUnclassified |
Guide to Pharmacology | None | None | None | None | 8702701 | |||
| 4514 | 3781 | 13 | None | -7 | 4 | Human | 7.8 | pIC50 | = | 7.8 | Functional | UnclassifiedUnclassified |
Guide to Pharmacology | None | None | None | None | 11602681 | |||
| 4514 | 3781 | 13 | None | -7 | 4 | Human | 7.8 | pIC50 | = | 7.8 | Functional | UnclassifiedUnclassified |
Guide to Pharmacology | None | None | None | None | 8702701 | |||
Showing 1 to 50 of 122 entries
| Ligands (move mouse cursor over ligand name to see structure) | Receptor | Assay information | Chemical information | |||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Sel. page | Similar- ity
| Common name
| GPCRdb ID | #Vendors
| Reference ligand | Fold selectivity | # Tested GPCRs
| Species | p-value (-log)
| Activity Type
| Activity Relation
| Activity Value
| Assay Type
| Assay Description
| Source | Mol weight | Rot Bonds | H don | H acc | LogP
| Smiles
| DOI |
Ligands (move mouse cursor over ligand name to see structure)
| Receptor
| Assay information
| Chemical information
| |||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sel. page | Similar- ity
| Common name
| GPCRdb ID | #Vendors
| Reference ligand | Fold selectivity | # Tested GPCRs
| Species | p-value (-log)
| Activity Type
| Activity Relation
| Activity Value
| Assay Type
| Assay Description
| Source | Mol weight | Rot Bonds | H don | H acc | LogP
| Smiles
| DOI |
| No data available in table | ||||||||||||||||||||||
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