Mutant Browser

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Protein name Generic number Position Segment Mutation FoldChange or Qual Exp Type Ligand Reference Review
p2y11_human 2.62x62 87 TM2 A => T N/A N/A Meis S et al (2010)
p2y11_human 6.55x55 268 TM6 R => A N/A N/A Meis S et al (2010)
Protein name Generic number Segment Position Mutation FoldChange or Qual Exp Type Ligand Reference Review


Residue

Diagrams

ICL1 K Q R P W ICL1ECL1 P K H W R Y ECL1ICL2 P F F A R S H L ICL2ECL2 H L K R P Q Q G A G N C S V A R P E A C I K C L G T A D H G ECL2ICL3 S P G M ICL3ECL3 W S T R C P S F A D I A Q A ECL3N-term M A A N V S G A K S C P A N F L A A A D D K L S G N-termC-term Y R D S W N P E D A K S T G Q A L P L N A T A A P K P S E P Q S R E L S Q C-term F Q G D F L W P I L V V E F L V A V A S N G L A L Y R F S I R H P A V V F S V Q L A V S D L L C A L T L P P L A A Y L Y P G E A A C R L E R F L F T C N L L G S V I F I T C I S L N R Y L G I V H R P K H A W A V S A A G W V L A A L L A M P T L S F S L A A Y R A Y S L V L A G L G C G L P L L L T L A A Y G A L G R A V L R T V A E K L R V A A L V A S G V A L Y A S S Y V P Y H I M R V L N V D A R R R T A A L E L G P Y V G Y Q V M R G L M P L A F C V H P L L Y M A A V P S C R H L G C C C P G
Download: PNG | SVG Increased binding/potency: >5-fold, >10-fold; Reduced binding/potency: >5-fold, >10-fold; No/low effect (<5-fold); and N/A
G N S A V A V L F E V V L I P W L F D G 1 V Q L A V S D L L C A L T L P P L A A Y 2 C T I F I V S G L L N C T F L F R E L R 3 A W A V S A A G W V L A A L L A M P T L 4 Y A A L T L L L P L G C G L G A L V L S Y 5 V A S G V A L Y S A S Y V P Y H I M R V L 6 L P H V C F A L P M L G R M V Q Y G V 7
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Residue Table


GPCRdb(A)
GPCRdb(A)
P2Y11 receptor
TM2
2x62 2.62x62 A87
TM6
6x55 6.55x55 R268